7-Nitro-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-tosyl-1H-indole is used as a reagent in the synthesis of piperazinyl pyrazolaminopyrimidinylindolylpropanamides as selective JAK1 inhibitors.
參考文獻
Aastrand, A. B. M., et al.: From PCT Int. Appl.?(2017),?WO?2017050938?A1?20170330